SCHEMBL7269755

SCHEMBL7269755

O=C(O)CCN1C(=O)CSc2ccccc21

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.63
KMT2A Q03164 3/20 0.63
LMNA P02545 2/20 0.63
NPSR1 Q6W5P4 1/20 0.56
TSHR P16473 2/20 0.53
ALDH1A1 P00352 2/20 0.53
CHRM1 P11229 1/20 0.52
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
ALOX15 P16050 1/20 0.47
GFER P55789 1/20 0.46
MAPT P10636 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5112508 0.86 MEN1 (0.60) MEN1KMT2ALMNAMMEACE
SCHEMBL4971618 0.85 NPSR1 (0.67) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL30808619 0.85 NPSR1 (0.67) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL7280026 0.83 NPSR1 (0.62) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL30808640 0.81 KMO (0.55) MEN1KMT2ALMNATSHRMAPT
SCHEMBL30808610 0.81 KMO (0.58) MEN1KMT2ALMNANPSR1ALDH1A1
SCHEMBL30808599 0.81 TSHR (0.46) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL9850726 0.81 NPSR1 (0.50) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL30808648 0.80 MEN1 (0.63) MEN1KMT2ALMNANPSR1TSHR
SCHEMBL12963502 0.80 NPSR1 (0.60) LMNANPSR1TSHRALDH1A1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023250002-A1 IDENTIFICATION OF NOVEL BENZOTHIAZONES AS TAU-SH3 INTERACTION INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE SOUTHERN RESEARCH INSTITUTE (US) 2023-12-28 WO disclosed
EP-0411751-A1 Renin inhibitory peptides Beecham Group p.l.c. (GB) 1991-02-06 EP disclosed