SCHEMBL7270294

SCHEMBL7270294

CC(C)C[C@H](NCCCNC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.59
CAPN2 P17655 1/20 0.59
HTT P42858 1/20 0.56
CTSK P43235 4/20 0.55
CTSS P25774 2/20 0.55
CTSL P07711 1/20 0.55
CTSB P07858 1/20 0.55
FOLH1 Q04609 1/20 0.55
CPB1 P15086 1/20 0.53
CPB2 Q96IY4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270291 1.00 CAPN1 (0.59) CAPN1CAPN2HTTCTSKCTSS
SCHEMBL7268833 0.92 HTT (0.55) CAPN1CAPN2HTTCTSKCTSS
SCHEMBL7268829 0.92 HTT (0.55) CAPN1CAPN2HTTCTSKCTSS
SCHEMBL7209805 0.86 HTT (0.64) HTTFOLH1
SCHEMBL11130487 0.83 SLC1A3 (0.57) CAPN1CAPN2CTSKCTSSCTSL
SCHEMBL5869834 0.83 SLC1A3 (0.57) CAPN1CAPN2CTSKCTSSCTSL
SCHEMBL5869839 0.83 SLC1A3 (0.57) CAPN1CAPN2CTSKCTSSCTSL
SCHEMBL5869829 0.83 SLC1A3 (0.57) CAPN1CAPN2CTSKCTSSCTSL
SCHEMBL7206127 0.82 HTT (0.59) HTTFOLH1
SCHEMBL6703436 0.82 CTSK (0.62) CAPN1CAPN2CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed