SCHEMBL7270587

SCHEMBL7270587

C=CC1OC(C)(C)N(C(=O)OC(C)(C)C)C1Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 8/20 0.41
KLK5 Q9Y337 7/20 0.39
CYP3A4 P08684 4/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 1/20 0.39
PRSS1 P07477 3/20 0.38
PRSS2 P07478 3/20 0.38
PRSS3 P35030 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ABCB1 P08183 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
PLA2G10 O15496 1/20 0.35
PLA2G5 P39877 1/20 0.35
STS P08842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2175304 0.91 KLK7 (0.40) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7962411 0.91 KLK7 (0.40) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL5833363 0.91 KLK7 (0.40) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL2175307 0.91 KLK7 (0.40) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7270193 0.87 KLK7 (0.38) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7270189 0.87 KLK7 (0.38) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7279540 0.87 KLK7 (0.38) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7279530 0.87 KLK7 (0.38) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL7950824 0.86 KLK7 (0.37) KLK7KLK5CYP3A4ALDH1A1MAPT
SCHEMBL9842063 0.85 KLK7 (0.41) KLK7KLK5CYP3A4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed