SCHEMBL7271372

SCHEMBL7271372

O=C(Cl)[C@@H]1CC[C@H]1C(=O)Cl

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 1/20 0.35
EPHX1 P07099 1/20 0.31
SLC1A2 P43004 2/20 0.31
SLC1A1 P43005 2/20 0.31
CYP2D6 P10635 2/20 0.30
LMNA P02545 2/20 0.30
BLM P54132 2/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
RAB9A P51151 1/20 0.30
MEN1 O00255 1/20 0.30
THRB P10828 1/20 0.30
PMP22 Q01453 1/20 0.30
KMT2A Q03164 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17237823 1.00 GABRR1 (0.35) GABRR1EPHX1SLC1A2SLC1A1CYP2D6
SCHEMBL2266700 1.00 GABRR1 (0.35) GABRR1EPHX1SLC1A2SLC1A1CYP2D6
SCHEMBL8191588 0.89 EPHX1 (0.40) EPHX1BLMTSHRRAB9AMEN1
SCHEMBL895753 0.89 EPHX1 (0.40) EPHX1BLMTSHRRAB9AMEN1
SCHEMBL11199858 0.89 EPHX1 (0.40) EPHX1BLMTSHRRAB9AMEN1
SCHEMBL7857943 0.89 PEPD (0.36) GABRR1EPHX1BLMMEN1KMT2A
SCHEMBL11199862 0.89 EPHX1 (0.40) EPHX1BLMTSHRRAB9AMEN1
SCHEMBL4744040 0.83
SCHEMBL22546037 0.83
SCHEMBL4812482 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111111475-B Preparation method of graphene oxide modified triptycenyl polyamide separation membrane 南京工业大学 2022-03-22 CN claimed
EP-3323500-B1 MANUFACTURING METHOD FOR TRIPTYCENE POLYMER CARRIER FILM NANJING UNIVERSITY OF TECHNOLOGY (CN) 2021-01-27 EP claimed
US-10799836-B2 Preparation method for triptyl polymer separation membrane NANJING TECH UNIVERSITY (CN) 2020-10-13 US claimed
CN-111111475-A Preparation method of graphene oxide modified triptycenyl polyamide separation membrane 南京工业大学 2020-05-08 CN claimed
US-20180236408-A1 A PREPARATION METHOD FOR TRIPTYL POLYMER SEPARATION MEMBRANE NANJING TECH UNIVERSITY (CN) 2018-08-23 US claimed
EP-3323500-A1 MANUFACTURING METHOD FOR TRIPTYCENE POLYMER CARRIER FILM Nanjing Tech University (CN) 2018-05-23 EP claimed
CN-111111475-B Preparation method of graphene oxide modified triptycenyl polyamide separation membrane 南京工业大学 2022-03-22 CN disclosed
EP-3323500-B1 MANUFACTURING METHOD FOR TRIPTYCENE POLYMER CARRIER FILM NANJING UNIVERSITY OF TECHNOLOGY (CN) 2021-01-27 EP disclosed
US-10799836-B2 Preparation method for triptyl polymer separation membrane NANJING TECH UNIVERSITY (CN) 2020-10-13 US disclosed
CN-111111475-A Preparation method of graphene oxide modified triptycenyl polyamide separation membrane 南京工业大学 2020-05-08 CN disclosed
US-10604536-B2 Substituted cyclopropanes as PDE-10 inhibitors Sunovion Pharamaceuticals Inc. (US) 2020-03-31 US disclosed
EP-2861596-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2019-03-20 EP disclosed
US-20180258104-A1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF Sunovion Pharamaceuticals Inc. 2018-09-13 US disclosed
WO-1996033159-A1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LABORATORIES (US) 1996-10-24 WO disclosed
US-5532372-A Imide derivatives, and their production and use SUMITOMO PHARMACEUTICALS COMPANY, LTD. (JP) 1996-07-02 US disclosed
US-5502075-A Leukotriene-B4 derivatives, process for their production and their use as pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1996-03-26 US disclosed
WO-1995004732-A1 OLIGOPEPTIDE ANTIRETROVIRAL AGENTS SYNPHAR LABORATORIES, INC. (CA) 1995-02-16 WO disclosed
WO-1992013838-A1 OLIGOPEPTIDE ANTIRETROVIRAL AGENTS SYNPHAR LABORATORIES, INC. (CA) 1992-08-20 WO disclosed
EP-0464846-A1 Imide derivatives, and their production and use SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1992-01-08 EP disclosed
US-5023335-A Antitumor agents ASTA PHARMA AKTIENGESELLSCHAFT 1991-06-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180258104-A1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF COMT, GPR119, NLN GABRR1 314/4885EPHX1 1105/4885SLC1A2 517/4885
US-10604536-B2 Substituted cyclopropanes as PDE-10 inhibitors PDE10A, PDE2A, PDE3A GABRR1 435/4885EPHX1 682/4885SLC1A2 2362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.