SCHEMBL7271671

SCHEMBL7271671

COc1ccc(CCNCCC=CCCNCCc2ccccc2)cc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.64
SIGMAR1 Q99720 2/20 0.63
ADRB2 P07550 2/20 0.58
DRD2 P14416 1/20 0.58
DRD1 P21728 1/20 0.58
DRD4 P21917 1/20 0.58
DRD3 P35462 1/20 0.58
POLB P06746 2/20 0.55
ATM Q13315 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
ALDH1A1 P00352 3/20 0.54
ALOX15 P16050 1/20 0.54
BCHE P06276 2/20 0.54
PLAAT3 P53816 1/20 0.54
PLAAT5 Q96KN8 1/20 0.54
PLAAT2 Q9NWW9 1/20 0.54
PLAAT4 Q9UL19 1/20 0.54
HTT P42858 3/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7271665 1.00 SLC2A1 (0.64) SLC2A1SIGMAR1ADRB2DRD2DRD1
SCHEMBL515430 0.91 SLC2A1 (0.74) SLC2A1SIGMAR1ADRB2DRD2DRD1
Bromide SCHEMBL11515734 0.90 SLC2A1 (0.72) SLC2A1SIGMAR1ADRB2DRD2DRD1
SCHEMBL27849455 0.86 SLC2A1 (0.85) SLC2A1SIGMAR1ADRB2DRD2DRD1
Hydrochloric Acid SCHEMBL7272231 0.84 SLC2A1 (0.87) SLC2A1SIGMAR1ADRB2DRD2DRD1
Hydrochloric Acid SCHEMBL7282863 0.84 SLC2A1 (0.70) SLC2A1SIGMAR1ADRB2DRD2DRD1
Hydrochloric Acid SCHEMBL10452455 0.84 SLC2A1 (0.87) SLC2A1SIGMAR1ADRB2DRD2DRD1
SCHEMBL7279400 0.84 ALDH1A1 (0.72) SLC2A1SIGMAR1ADRB2SMN1; SMN2ALDH1A1
SCHEMBL13344551 0.84 SLC2A1 (0.87) SLC2A1SIGMAR1ADRB2DRD2DRD1
SCHEMBL7435099 0.83 ATM (0.76) SLC2A1SIGMAR1ADRB2POLBATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375668-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1990-06-27 EP disclosed
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed