SCHEMBL7271817

SCHEMBL7271817

C/C(N)=C\c1nc(-c2ccccc2)cs1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
ATP4A P20648 1/20 0.50
ATP4B P51164 1/20 0.50
KMT2A Q03164 7/20 0.49
MEN1 O00255 6/20 0.49
MAPT P10636 5/20 0.49
LMNA P02545 4/20 0.49
KDM4E B2RXH2 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
NFKB1 P19838 1/20 0.49
RAB9A P51151 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
CYP3A4 P08684 1/20 0.49
GAA P10253 3/20 0.48
GFER P55789 2/20 0.47
ALOX12 P18054 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.44
SREBF2 Q12772 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7271819 1.00 ALDH1A1 (0.51) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL16402070 0.85 MAPT (0.47) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL4573806 0.79 ALDH1A1 (0.53) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL4573034 0.78 ALDH1A1 (0.55) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL15401707 0.75 PARP1 (0.49) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL15401706 0.75 PARP1 (0.49) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL10622090 0.74 ALDH1A1 (0.55) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL2224538 0.74 ALDH1A1 (0.55) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL27660527 0.74 ALDH1A1 (0.55) ALDH1A1ATP4AATP4BKMT2AMEN1
SCHEMBL3698383 0.73 MEN1 (0.45) ALDH1A1ATP4AATP4BKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4760147-A Isopropyl 1,4-dihydro-2,6-dimethyl-4-(2,3-dichlorophenyl)-3-(1,3,4-oxadiazol-2 -yl)pyridine-5-carboxylate CASSELLA AKTIENGESELLSCHAFT (DE) 1988-07-26 US disclosed
EP-0172509-A2 Process for the preparation of optically active, substituted 1,4-dihydropyridines and their use as medicaments CASSELLA Aktiengesellschaft (DE) 1986-02-26 EP disclosed
US-4558058-A HYPOTENSIVE AGENTS CASSELLA AKTIENGESELLSCHAFT (DE) 1985-12-10 US disclosed
EP-0116708-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use as pharmaceuticals CASSELLA Aktiengesellschaft (DE) 1984-08-29 EP disclosed