SCHEMBL7272913

SCHEMBL7272913

COCCOC(=O)OC1=C(C)NC(C)=C(c2nnco2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.46
CYP2C9 P11712 3/20 0.46
KDM4E B2RXH2 3/20 0.46
ABCB11 O95342 3/20 0.46
TBXA2R P21731 3/20 0.46
ADRA1A P35348 3/20 0.46
SLC6A3 Q01959 3/20 0.46
MEN1 O00255 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
HIF1A Q16665 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
TSHR P16473 2/20 0.46
ABCB1 P08183 2/20 0.46
ADORA3 P0DMS8 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10866129 0.92 KMT2A (0.45) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL10870367 0.90 ALDH1A1 (0.43) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL7272930 0.90 KMT2A (0.45) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL10620583 0.88 CYP2C9 (0.56) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL10867143 0.88 KDM4E (0.42) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL7273136 0.86 ALDH1A1 (0.41) KMT2ACYP2C9KDM4ECYP3A4CYP2C19
SCHEMBL10862617 0.86 KMT2A (0.42) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL7263830 0.86 CYP2C9 (0.39) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL10868478 0.85 CYP2C9 (0.44) KMT2ACYP2C9KDM4EABCB11TBXA2R
SCHEMBL10864909 0.85 CYP2C9 (0.44) KMT2ACYP2C9KDM4EABCB11TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0172509-A2 Process for the preparation of optically active, substituted 1,4-dihydropyridines and their use as medicaments CASSELLA Aktiengesellschaft (DE) 1986-02-26 EP disclosed
EP-0116708-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use as pharmaceuticals CASSELLA Aktiengesellschaft (DE) 1984-08-29 EP disclosed