SCHEMBL7273464

SCHEMBL7273464

N#Cc1ccc(-c2ccc(Nc3ncccc3N)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
ABCG2 Q9UNQ0 6/20 0.50
PDE10A Q9Y233 1/20 0.47
IKBKB O14920 1/20 0.46
HPGD P15428 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP11B2 P19099 1/20 0.44
DHODH Q02127 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4807750 0.95 CA12 (0.57) CA12CA1CA2CA9ABCG2
SCHEMBL6797398 0.79 ABCG2 (0.56) CA12CA1CA2CA9ABCG2
SCHEMBL7695744 0.79 CA12 (0.68) CA12CA1CA2CA9PDE10A
SCHEMBL23319512 0.77 ABCG2 (0.50) ABCG2HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL10094595 0.77 NPC1 (0.51) ABCG2HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL2472176 0.77 JAK2 (0.40) CA12CA1CA2CA9ABCG2
SCHEMBL19851118 0.76 CA12 (0.63) CA12CA1CA2CA9ABCG2
SCHEMBL1859867 0.76 CA12 (0.63) CA12CA1CA2CA9ABCG2
SCHEMBL11394107 0.74 CA12 (0.62) CA12CA1CA2CA9PDE10A
SCHEMBL11398989 0.74 CA12 (0.62) CA12CA1CA2CA9ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed