SCHEMBL7274145

SCHEMBL7274145

Cc1c(-c2ccc(C(=N)N)cc2)n(-c2ccccc2)c(=O)n1-c1ccc(CCC(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.54
ITGA2B P08514 7/20 0.54
PLA2G4A P47712 1/20 0.43
FFAR1 O14842 2/20 0.42
F2 P00734 3/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40
TMPRSS15 P98073 1/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
F7 P08709 1/20 0.39
F3 P13726 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273934 1.00 ITGB3 (0.54) ITGB3ITGA2BPLA2G4AFFAR1F2
SCHEMBL7393913 0.90 ITGB3 (0.43) ITGB3ITGA2BF2F10PRSS1
SCHEMBL7391063 0.90 ITGB3 (0.43) ITGB3ITGA2BF2F10PRSS1
Hydrochloric Acid SCHEMBL7283228 0.89 ITGB3 (0.42) ITGB3ITGA2BF2F10PRSS1
Hydrochloric Acid SCHEMBL7284140 0.89 ITGB3 (0.42) ITGB3ITGA2BF2F10PRSS1
SCHEMBL7282771 0.88 ITGB3 (0.55) ITGB3ITGA2BPLA2G4AFFAR1F2
SCHEMBL7275237 0.88 ITGB3 (0.55) ITGB3ITGA2BPLA2G4AFFAR1F2
SCHEMBL7275218 0.81 NQO2 (0.42) ITGB3ITGA2BF2F7F3
SCHEMBL7274401 0.80 ITGB3 (0.55) ITGB3ITGA2BPLA2G4AFFAR1F2
SCHEMBL7282872 0.80 ITGB3 (0.55) ITGB3ITGA2BPLA2G4AFFAR1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587134-A2 Cyclic urea derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-03-16 EP claimed
US-5880284-A HAVING ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASES-INHIBITING EFFECTS DR. KARL THOMAE GMBH (DE) 1999-03-09 US disclosed
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5681841-A PREVENTION CELL AGGREGATION KARL THOMAE GMBH (DE) 1997-10-28 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
EP-0587134-A2 Cyclic urea derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-03-16 EP disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed