SCHEMBL7275804

SCHEMBL7275804

Cc1ccc(S(=O)(=O)NC(Cc2ccccc2)C(O)C(Cc2ccccc2)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.50
CA7 P43166 2/20 0.50
ALDH1A1 P00352 5/20 0.49
TSHR P16473 2/20 0.49
KLK5 Q9Y337 3/20 0.49
GAA P10253 1/20 0.48
CTSL P07711 2/20 0.47
MAPT P10636 1/20 0.46
ATM Q13315 1/20 0.46
MMP9 P14780 1/20 0.45
LMNA P02545 2/20 0.45
PKM P14618 2/20 0.45
HPGD P15428 2/20 0.45
HTT P42858 2/20 0.45
KMT2A Q03164 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
MEN1 O00255 1/20 0.45
ALOX15 P16050 1/20 0.45
XBP1 P17861 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270385 0.90 KLK5 (0.52) CA2CA7ALDH1A1TSHRKLK5
SCHEMBL7278016 0.85 CA2 (0.61) CA2CA7ALDH1A1GAACTSL
SCHEMBL9848360 0.84 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL7270592 0.84 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL6445261 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL8532202 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL6446193 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL6444857 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL8534875 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM
SCHEMBL6445320 0.82 KLK5 (0.63) ALDH1A1TSHRKLK5CTSLATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed