SCHEMBL7276534

SCHEMBL7276534

O=Cc1cc([N+](=O)[O-])ccc1SCCCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.47
CYP2C19 P33261 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 4/20 0.43
POLB P06746 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488789 0.97 CYP1A2 (0.48) HTR1ACYP2C19CYP1A2CYP2D6ALDH1A1
SCHEMBL9691023 0.80 MGAM (0.53) HTR1AALDH1A1GAA
SCHEMBL4960591 0.78 CYP2C19 (0.59) HTR1ACYP2C19CYP1A2CYP2D6ALDH1A1
SCHEMBL4962109 0.78 CYP1A2 (0.58) HTR1ACYP2C19CYP1A2CYP2D6ALDH1A1
SCHEMBL8395124 0.77 GSTP1 (0.50) CYP2C19CYP1A2ALDH1A1POLBMEN1
SCHEMBL8398603 0.77 ERN1 (0.46) ALDH1A1MEN1GAAKMT2A
SCHEMBL8399950 0.77 ERN1 (0.46) ALDH1A1MEN1GAAKMT2A
SCHEMBL4960929 0.73 MAPT (0.53) HTR1ACYP2C19CYP1A2CYP2D6ALDH1A1
SCHEMBL4963360 0.73 MAPT (0.53) HTR1ACYP2C19CYP1A2CYP2D6ALDH1A1
SCHEMBL7278367 0.72 CYP3A4 (0.49) ALDH1A1POLBMEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276552-A1 1,4-dihydropyridine derivatives and their production YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1988-08-03 EP claimed
US-5039674-A Calcium antagonistics YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-08-13 US disclosed
US-4782160-A CALCIUM RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-11-01 US disclosed
EP-0276552-A1 1,4-dihydropyridine derivatives and their production YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1988-08-03 EP disclosed