SCHEMBL7276958

SCHEMBL7276958

CC(C)(C)OC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ccc(C(=N)N)cn3)cc2)NC1=O

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.61
ITGA2B P08514 1/20 0.61
GPR119 Q8TDV5 3/20 0.38
RXFP1 Q9HBX9 1/20 0.34
CHEK2 O96017 2/20 0.34
IRAK4 Q9NWZ3 5/20 0.33
DGAT1 O75907 4/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7277321 0.99 ITGB3 (0.61) ITGB3ITGA2BGPR119RXFP1CHEK2
SCHEMBL7277517 0.91 ITGB3 (0.65) ITGB3ITGA2BGPR119RXFP1IRAK4
Hydrochloric Acid SCHEMBL7284744 0.90 ITGB3 (0.64) ITGB3ITGA2BRXFP1IRAK4DGAT1
Hydrochloric Acid SCHEMBL7277371 0.90 ITGB3 (0.61) ITGB3ITGA2BCHEK2IRAK4
SCHEMBL9261874 0.88 ITGB3 (0.61) ITGB3ITGA2BGPR119RXFP1IRAK4
Hydrochloric Acid SCHEMBL7285261 0.88 ITGB3 (0.61) ITGB3ITGA2BRXFP1IRAK4MAPT
Hydrochloric Acid SCHEMBL7287064 0.88 ITGB3 (0.57) ITGB3ITGA2BGPR119RXFP1IRAK4
SCHEMBL7277434 0.88 ITGB3 (0.80) ITGB3ITGA2BRXFP1IRAK4DGAT1
Hydrochloric Acid SCHEMBL7285424 0.87 ITGB3 (0.54) ITGB3ITGA2BGPR119IRAK4DGAT1
Hydrochloric Acid SCHEMBL7278436 0.85 ITGB3 (0.58) ITGB3ITGA2BRXFP1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed