SCHEMBL7277175

SCHEMBL7277175

COc1cc2c(cc1OC)CC(/C=N/O)=C2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
CYP3A4 P08684 1/20 0.42
BRD4 O60885 1/20 0.38
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 4/20 0.35
MAOA P21397 3/20 0.35
GLA P06280 2/20 0.35
ACHE P22303 4/20 0.34
KMT2A Q03164 2/20 0.33
NPC1 O15118 2/20 0.33
NFKB1 P19838 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
GFER P55789 1/20 0.32
GAA P10253 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277184 1.00 MAPT (0.42) MAPTCYP3A4BRD4ALDH1A1KDM4E
SCHEMBL7277292 1.00 MAPT (0.42) MAPTCYP3A4BRD4ALDH1A1KDM4E
SCHEMBL7274442 0.86 KDM4E (0.41) MAPTCYP3A4ALDH1A1KDM4EMAOA
SCHEMBL7269563 0.86 KDM4E (0.41) MAPTCYP3A4ALDH1A1KDM4EMAOA
SCHEMBL7269567 0.86 KDM4E (0.41) MAPTCYP3A4ALDH1A1KDM4EMAOA
SCHEMBL10710146 0.78 CYP3A4 (0.47) MAPTCYP3A4BRD4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL10709161 0.75 CYP3A4 (0.34) MAPTCYP3A4BRD4ACHE
SCHEMBL10711798 0.72 FDPS (0.41) MAPTCYP3A4BRD4ALDH1A1KDM4E
SCHEMBL10711789 0.72 FDPS (0.41) MAPTCYP3A4BRD4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL10714768 0.70 CYP3A4 (0.35) MAPTCYP3A4BRD4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352832-B1 COMPOUNDS WITH BRONCHODILATOR ACTIVITY AKZO N.V. (NL) 1992-05-06 EP disclosed
US-5026724-A Benzothiophene derivatives AKZO N.V. (NL) 1991-06-25 US disclosed
EP-0352832-A1 Compounds with bronchodilator activity AKZO N.V. (NL) 1990-01-31 EP disclosed