SCHEMBL7277206

SCHEMBL7277206

N=C(N)c1ccc(-c2ccc(OC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3c3ccccn3)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.55
ITGA2B P08514 6/20 0.55
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
SLC6A7 Q99884 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
F2 P00734 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34
TMPRSS6 Q8IU80 1/20 0.34
ST14 Q9Y5Y6 1/20 0.34
PPARD Q03181 2/20 0.34
FFAR4 Q5NUL3 1/20 0.34
FFAR1 O14842 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277743 0.91 ITGB3 (0.44) ITGB3ITGA2BALDH1A1MAPK1MEN1
SCHEMBL7275881 0.90 ITGB3 (0.59) ITGB3ITGA2BF2PRSS1PRSS2
Water SCHEMBL8882684 0.89 ITGB3 (0.58) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7287049 0.86 ITGB3 (0.53) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7274581 0.85 ITGB3 (0.58) ITGB3ITGA2BPRSS1
SCHEMBL7272584 0.85 ITGB3 (0.58) ITGB3ITGA2BPRSS1PARP10
SCHEMBL7275867 0.84 ITGB3 (0.55) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7281034 0.84 ITGB3 (0.55) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL7276861 0.84 ITGB3 (0.55) ITGB3ITGA2BF2PRSS1PPARD
SCHEMBL7281058 0.83 ITGB3 (0.54) ITGB3ITGA2BF2PRSS1PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP claimed
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed