SCHEMBL7277477

SCHEMBL7277477

C=CCOC(=O)NC(CC(=O)OC(C)(C)C)C(=O)CCCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 18/20 0.60
ALDH1A1 P00352 1/20 0.44
ACE P12821 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277471 0.97 CASP1 (0.59) CASP1ALDH1A1ACE
SCHEMBL7286909 0.94 CASP1 (0.65) CASP1ALDH1A1ACE
SCHEMBL5832716 0.88 CASP1 (0.56) CASP1ALDH1A1
SCHEMBL7486694 0.86 CASP1 (0.77) CASP1
SCHEMBL7286930 0.83 CASP1 (0.52) CASP1ALDH1A1
SCHEMBL7286618 0.81 CASP1 (0.48) CASP1ALDH1A1
SCHEMBL7275372 0.80 CASP1 (0.48) CASP1ALDH1A1
SCHEMBL7278924 0.80 CASP1 (0.47) CASP1
SCHEMBL2801332 0.79 CASP1 (0.54) CASP1
SCHEMBL12450829 0.79 CASP1 (0.53) CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519748-B1 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO INC (US) 1998-09-02 EP disclosed
US-5434248-A Peptidyl derivatives as inhibitors of interleukin-1β converting enzyme MERCK & CO., INC. (US) 1995-07-18 US disclosed
EP-0519748-A2 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO. INC. (US) 1992-12-23 EP disclosed