SCHEMBL7278375

SCHEMBL7278375

O=c1c2c(ncn2Cc2cccc(Br)c2)c2cccnc2n1-c1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.80
PDE4B Q07343 6/20 0.66
PDE4C Q08493 6/20 0.66
PDE4D Q08499 6/20 0.66
PDE1A P54750 1/20 0.47
PDE1B Q01064 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.41
FEN1 P39748 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
YTHDC1 Q96MU7 1/20 0.40
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272788 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7278584 0.88 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7280079 0.86 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7278166 0.85 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7270989 0.85 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL29416766 0.85 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL2278414 0.85 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7271034 0.84 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7281912 0.83 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL7271255 0.82 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DPDE1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459505-B1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-10-02 EP disclosed
US-5536730-A ANTIINFLAMMATORY, ANTIALLERGIC AND BRONCHODILATIVE ACTIVITY KYOWA HAKKO KOGYO CO. LTD. (JP) 1996-07-16 US disclosed
US-5468756-A Antiinflammatory, antiallergen KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-21 US disclosed
US-5364859-A Antiinflammatory agents, antiallergens, bronchodilators KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-11-15 US disclosed
EP-0459505-A1 Imidazonaphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-04 EP disclosed