SCHEMBL7278459

SCHEMBL7278459

CCCCSc1ccc(-c2nc3cnccc3[nH]2)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 7/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
AR P10275 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
CYP1A2 P05177 4/20 0.39
CYP2E1 P05181 4/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2C8 P10632 4/20 0.39
CYP2D6 P10635 4/20 0.39
CYP2C9 P11712 4/20 0.39
CYP2B6 P20813 4/20 0.39
CYP2C19 P33261 4/20 0.39
AMY1A P0DUB6 3/20 0.38
AAK1 Q2M2I8 1/20 0.38
PDE2A O00408 1/20 0.36
CDK4 P11802 1/20 0.36
CCNA2 P20248 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7271872 0.94 PDE5A (0.48) PDE5APDE3BPDE3AARKDM4E
SCHEMBL7281156 0.91 PDE5A (0.48) PDE5APDE3BPDE3AARKDM4E
SCHEMBL7272787 0.89 PDE5A (0.50) PDE5APDE3BPDE3AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7270687 0.88 PDE5A (0.50) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL7279533 0.84 PDE5A (0.45) PDE5APDE3BPDE3AARKDM4E
SCHEMBL7271721 0.83 PDE5A (0.53) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL9634871 0.83 PDE5A (0.47) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL9635715 0.83 PDE5A (0.47) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL9634366 0.83 PDE5A (0.47) PDE5APDE3BPDE3AKDM4EALDH1A1
SCHEMBL9636125 0.82 PDE5A (0.48) PDE5APDE3BPDE3AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904785-A INOTROPIC AGENTS FOR CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1990-02-27 US disclosed
US-4758574-A 2-phenylimidazio (4,5-c) pyridines ELI LILLY AND COMPANY (US) 1988-07-19 US disclosed
EP-0093593-A2 Pyridine compounds ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed