SCHEMBL7279533

SCHEMBL7279533

CCCSc1ccc(-c2nc3cnccc3[nH]2)c(OCC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 11/20 0.45
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNH2 Q12809 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PDE10A Q9Y233 2/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
GUSB P08236 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
PDE4A P27815 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281156 0.94 PDE5A (0.48) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL7272133 0.91 PDE5A (0.42) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL7271872 0.90 PDE5A (0.48) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL7278432 0.88 PDE5A (0.43) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL7278459 0.84 PDE5A (0.47) PDE5APDE3BPDE3AHPGDCYP1A2
SCHEMBL7272842 0.84 PDE5A (0.50) PDE5APDE3BPDE3ANPSR1KDM4E
SCHEMBL7279872 0.82 CBFB (0.46) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL7280960 0.82 PDE5A (0.45) PDE5APDE3BPDE3ASMN1; SMN2PDE10A
SCHEMBL7272787 0.81 PDE5A (0.50) PDE5APDE3BPDE3AHPGDSMN1; SMN2
SCHEMBL9635782 0.81 PDE5A (0.44) PDE5APDE3BPDE3AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904785-A INOTROPIC AGENTS FOR CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1990-02-27 US disclosed
US-4758574-A 2-phenylimidazio (4,5-c) pyridines ELI LILLY AND COMPANY (US) 1988-07-19 US disclosed
EP-0093593-A2 Pyridine compounds ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed