SCHEMBL7279331

SCHEMBL7279331

CC(C)N1C(=O)C(O)N(O)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
AADAT Q8N5Z0 3/20 0.35
XIAP P98170 2/20 0.34
ALDH1A1 P00352 4/20 0.33
P2RX4 Q99571 2/20 0.33
P2RX1 P51575 1/20 0.33
P2RX3 P56373 1/20 0.33
P2RX7 Q99572 1/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
ALOX15 P16050 1/20 0.33
GOT1 P17174 1/20 0.33
BCHE P06276 1/20 0.33
KYAT1 Q16773 1/20 0.33
KYAT3 Q6YP21 1/20 0.33
RAD52 P43351 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4415567 0.74 SMN1; SMN2 (0.42) CYP2D6CYP2C9SMN1; SMN2AADATXIAP
SCHEMBL30396025 0.70 SMN1; SMN2 (0.46) CYP2D6CYP2C9SMN1; SMN2ALDH1A1P2RX4
SCHEMBL5000976 0.70 SMN1; SMN2 (0.46) CYP2D6CYP2C9SMN1; SMN2ALDH1A1P2RX4
SCHEMBL7324240 0.67 MEN1 (0.57) CYP2C9SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL38660167 0.67 ALDH1A1 (0.41) CYP2D6CYP2C9SMN1; SMN2AADATXIAP
SCHEMBL28227456 0.67 ALDH1A1 (0.41) CYP2D6CYP2C9SMN1; SMN2AADATXIAP
SCHEMBL4422532 0.66 CYP2D6 (0.58) CYP2D6CYP2C9SMN1; SMN2AADATXIAP
SCHEMBL4422526 0.66 CYP2D6 (0.58) CYP2D6CYP2C9SMN1; SMN2AADATXIAP
SCHEMBL4415354 0.66 SMN1; SMN2 (0.57) CYP2D6CYP2C9SMN1; SMN2ALDH1A1MEN1
SCHEMBL7688831 0.66 SMN1; SMN2 (0.57) CYP2D6CYP2C9SMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320136-B1 Imidazoquinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-07-27 EP disclosed
US-4999354-A Central Nervous System Disorders, Anticonvulsant and Anxiolytic Agents A/S FERROSAN (DK) 1991-03-12 US disclosed
US-4968682-A CENTRAL NERVOUS SYSTEM DISORDERS A/S FERROSAN (DK) 1990-11-06 US disclosed
EP-0320136-A2 Imidazoquinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1989-06-14 EP disclosed