SCHEMBL7279809

SCHEMBL7279809

CC(C)(C)NC(=O)[C@@H]1C[C@H](OCc2ccccc2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.51
MCL1 Q07820 11/20 0.47
KLK7 P49862 1/20 0.46
HTRA1 Q92743 1/20 0.43
MMP9 P14780 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
GHSR Q92847 2/20 0.42
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945215 0.90 ABCB1 (0.51) ABCB1MCL1KLK7HTRA1MMP9
SCHEMBL6945211 0.90 ABCB1 (0.51) ABCB1MCL1KLK7HTRA1MMP9
SCHEMBL26604823 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL7287734 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL708629 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL949983 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL1448119 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL3179881 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL376159 0.88 ABCB1 (0.52) ABCB1MCL1KLK7
SCHEMBL708630 0.88 ABCB1 (0.52) ABCB1MCL1KLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552405-A TREATMENT OF AIDS, ACTIVITY AGAINST RETROVIRUSES BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH, INC. (CA) 1996-09-03 US disclosed
EP-0560269-B1 Substituted pyrrolidine derivatives as HIV protease inhibitors BIO MEGA BOEHRINGER INGELHEIM (CA) 1995-05-31 EP disclosed
EP-0560269-A1 Substituted pyrrolidine derivatives as HIV protease inhibitors BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1993-09-15 EP disclosed