SCHEMBL7279844

SCHEMBL7279844

NC(=O)c1cccc2c1OCC(=O)N2

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.60
PARP1 P09874 5/20 0.56
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.40
CREBBP Q92793 2/20 0.39
BRD4 O60885 1/20 0.39
SCN5A Q14524 2/20 0.39
SCN9A Q15858 2/20 0.39
AURKA O14965 1/20 0.39
RAF1 P04049 1/20 0.38
BRAF P15056 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
SCN1A P35498 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7373686 0.98 SMYD3 (0.58) SMYD3PARP1GAAKMT2ACREBBP
SCHEMBL31364686 0.86 SMYD3 (0.57) SMYD3PARP1GAAKMT2ACREBBP
SCHEMBL306669 0.86 SMYD3 (0.57) SMYD3PARP1GAAKMT2ACREBBP
SCHEMBL17476309 0.84 SMYD3 (0.56) SMYD3PARP1GAAKMT2ACREBBP
SCHEMBL29753562 0.81 SMYD3 (0.56) SMYD3GAAKMT2ACREBBPBRD4
SCHEMBL1340605 0.81 SMYD3 (0.56) SMYD3GAAKMT2ACREBBPBRD4
SCHEMBL17476304 0.81 SMYD3 (0.56) SMYD3GAAKMT2ACREBBPBRD4
SCHEMBL6181892 0.77 SMYD3 (0.50) SMYD3PARP1GAACREBBPBRD4
SCHEMBL4317646 0.77 SMYD3 (0.51) SMYD3PARP1GAACREBBPBRD4
SCHEMBL254031 0.77 SMYD3 (0.48) SMYD3PARP1KMT2ACREBBPBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1262548-C Synthesis of benzoxazine monohydrochlorate compound XINYI WANXIANG PHARMACEUTICAL (CN) 2006-07-05 CN disclosed
CN-1552699-A Synthesis of benzoxazine monohydrochlorate compound 上海延安万象药业股份有限公司 2004-12-08 CN disclosed
EP-0407137-B1 Benzazine compounds and pharmaceutical uses thereof YOSHITOMI PHARMACEUTICAL (JP) 1996-05-01 EP disclosed
US-5185333-A Dopamine D2 receptor blocking agents YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1993-02-09 US disclosed
EP-0407137-A2 Benzazine compounds and pharmaceutical uses thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-01-09 EP disclosed