SCHEMBL7280455

SCHEMBL7280455

O=C1COc2c(cc(Cl)cc2C(=O)NC2CN3CCC2CC3)N1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.65
KCNH2 Q12809 2/20 0.65
HTR2A P28223 1/20 0.65
SLC6A4 P31645 1/20 0.65
HRH1 P35367 1/20 0.65
PDE4D Q08499 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
CYP1A2 P05177 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7281902 0.99 HTR3A (0.64) HTR3AKCNH2HTR2ASLC6A4HRH1
SCHEMBL7268990 0.82 HTR3A (0.69) HTR3AKCNH2HTR2ASLC6A4HRH1
SCHEMBL31387673 0.82 HTR3A (0.58) HTR3AKCNH2HTR2ASLC6A4HRH1
SCHEMBL7289440 0.82 HTR3A (0.58) HTR3AKCNH2HTR2ASLC6A4HRH1
Hydrochloric Acid SCHEMBL7276091 0.82 HTR3A (0.68) HTR3AKCNH2HTR2ASLC6A4HRH1
Hydrochloric Acid SCHEMBL7289083 0.81 HTR3A (0.57) HTR3AKCNH2HTR2ASLC6A4HRH1
Azasetron SCHEMBL19492326 0.79 HTR3A (1.00) HTR3AKCNH2HTR2ASLC6A4HRH1
Azasetron SCHEMBL17191 0.79 HTR3A (1.00) HTR3AKCNH2HTR2ASLC6A4HRH1
Azasetron SCHEMBL29880168 0.79 HTR3A (1.00) HTR3AKCNH2HTR2ASLC6A4HRH1
Azasetron SCHEMBL19463750 0.79 HTR3A (1.00) HTR3AKCNH2HTR2ASLC6A4HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0313393-B1 Benzoxazine compounds and pharmaceutical use thereof YOSHITOMI PHARMACEUTICAL (JP) 1994-03-16 EP disclosed
US-4892872-A ANTIEMETICS, ANTINAUSEA YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed
EP-0313393-A2 Benzoxazine compounds and pharmaceutical use thereof Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-04-26 EP disclosed