SCHEMBL7282255

SCHEMBL7282255

COc1ccccc1NC(=O)CN1CCN(CC(O)COc2ccccc2OC)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.76
CYP2D6 P10635 3/20 0.76
CYP3A4 P08684 2/20 0.76
NFKB1 P19838 1/20 0.76
ADRB2 P07550 1/20 0.76
ADRB1 P08588 1/20 0.76
ADRA2A P08913 1/20 0.76
ADRA2B P18089 1/20 0.76
ADRA2C P18825 1/20 0.76
ADRA1A P35348 1/20 0.76
DRD3 P35462 1/20 0.76
HTR2B P41595 1/20 0.76
KCNH2 Q12809 1/20 0.76
SCN5A Q14524 1/20 0.76
NPSR1 Q6W5P4 5/20 0.74
LMNA P02545 2/20 0.74
BLM P54132 1/20 0.74
PMP22 Q01453 1/20 0.74
ALDH1A1 P00352 6/20 0.64
KMT2A Q03164 7/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10837597 0.92 TSHR (0.71) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL4867116 0.90 CYP3A4 (0.71) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7282511 0.89 CYP3A4 (0.86) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7291659 0.89 CYP2D6 (0.76) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7279455 0.89 CYP3A4 (0.67) TSHRCYP2D6CYP3A4NFKB1ADRB2
Hydrochloric Acid SCHEMBL7300686 0.88 LMNA (0.76) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7288476 0.88 TSHR (0.74) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7279519 0.87 CYP3A4 (0.76) TSHRCYP2D6CYP3A4NFKB1ADRB2
SCHEMBL7281999 0.87 TSHR (0.73) TSHRCYP2D6CYP3A4NFKB1ADRB2
Ranolazine SCHEMBL7933344 0.86 CYP3A4 (1.00) TSHRCYP2D6CYP3A4NFKB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed