SCHEMBL72823

SCHEMBL72823

O=C1OC(=O)c2cc(C#Cc3ccccc3)ccc21

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 15/20 0.66
ALOX15 P16050 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
APP P05067 1/20 0.46
HNF4A P41235 1/20 0.43
MAPT P10636 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9611211 0.94 GRM5 (0.56) GRM5ALOX15TDP1ALDH1A1
SCHEMBL2640689 0.92 GRM5 (0.53) GRM5ALOX15TDP1ALDH1A1
Toluene SCHEMBL7860098 0.92 GRM5 (0.57) GRM5ALOX15TDP1
SCHEMBL9885475 0.91 GRM5 (0.56) GRM5ALOX15TDP1MAPTALDH1A1
SCHEMBL3447309 0.87 GRM5 (0.51) GRM5ALOX15TDP1APPMAPT
SCHEMBL14357420 0.86 GRM5 (0.58) GRM5APP
SCHEMBL9885466 0.86 GRM5 (0.54) GRM5APPHNF4A
SCHEMBL9885459 0.85 GRM5 (0.49) GRM5ALOX15TDP1ALDH1A1
SCHEMBL27186006 0.85 GRM5 (0.49) GRM5ALOX15TDP1MAPTALDH1A1
SCHEMBL4577919 0.85 GRM5 (0.49) GRM5ALOX15TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2720 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119613717-B Thermosetting polyimide resin with high heat resistance and preparation method thereof SICHUAN UNIVERSITY (CN) 2026-05-26 CN claimed
CN-122080070-A Ionic liquid flame retardant, epoxy resin composite material, and preparation method and application thereof 2026-05-26 CN claimed
CN-122080406-A High-temperature-resistant and thermally-dimensionally-stable soluble polyimide resin and preparation method and application thereof 2026-05-26 CN claimed
WO-2026102770-A1 CROSS-LINKED POLYIMIDE LITHIUM BATTERY SEPARATOR, PREPARATION METHOD THEREFOR AND USE THEREOF 亚安顶材有限公司 2026-05-21 WO claimed
WO-2026099626-A1 METHODS AND SYSTEMS FOR MANUFACTURING RADIOPHARMACEUTICALS NOVARTIS AG (CH) 2026-05-15 WO claimed
WO-2026098441-A1 COMPOSITION AND METHOD FOR CANCER TREATMENT USING POLYPEPTIDE CONJUGATES SUZHOU SMARTNUCLIDE BIOPHARMACEUTICAL CO., LTD. (CN) 2026-05-15 WO claimed
CN-122005879-A Modified GRPR antagonist peptides for cancer imaging and treatment 慕尼黑工业大学 2026-05-12 CN claimed
EP-4735055-A1 UROKINASE-TYPE PLASMINOGEN ACTIVATOR RECEPTOR (UPAR)-PET/CT IN BRAIN TUMOURS Curasight A/S (DK) 2026-05-06 EP claimed
US-20260077071-A1 Targeted Delivery of Theranostic Agents PETER MACCALLUM CANCER INST (AU) 2026-03-19 US claimed
US-20260048156-A1 FAP-TARGETING PHARMACEUTICAL PRODUCT FOR THERAPY AND DIAGNOSIS OF CANCERS Atoms for Cure GmbH (DE) 2026-02-19 US claimed
US-6124035-A High temperature transfer molding resins THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 2000-09-26 US claimed
EP-1018507-A1 Terminal-modified imide oligomers and cured products thereof Ube Industries, Ltd. (JP) 2000-07-12 EP claimed
US-6084106-A Adhesion promoters and methods of their synthesis and use THIOKOL CORPORATION (US) 2000-07-04 US claimed
EP-1000108-A1 AQUEOUS POLYIMIDE PROCESS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-05-17 EP claimed
WO-1999062989-A1 FILMS, PREIMPREGNATED TAPES AND COMPOSITES MADE FROM POLYIMIDE 'SALT-LIKE' SOLUTIONS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (NASA) (US) 1999-12-09 WO claimed
WO-1999006470-A1 AQUEOUS POLYIMIDE PROCESS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1999-02-11 WO claimed
US-5681967-A ENDCAPPING POLYAMIC ACIDS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1997-10-28 US claimed
US-5644022-A ENDCAPPING THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMNINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1997-07-01 US claimed
US-5567800-A MOLECULAR WEIGHT CONTROLLED AROMATIC POLYIMIDES; ELONGATION, HIGH GLASS TRANSITION TEMPERATURE, TOUGHNESS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE ADMINISTRATOR OF THE NATIONAL AERONAUTICS AND SPACE ADMINISTRATION (US) 1996-10-22 US claimed
US-5478913-A Copolymerizing biphenyl dianhydride as ester/acid/ with mix of m- or p-phenylenediamines and aminophenoxybenzene component encapped with phthalic anhydride or ethynyl-group amine or anhydride; heat, oxidation resistant; prepregs E. I. DU PONT DE NEMOURS AND COMPANY (US) 1995-12-26 US claimed