SCHEMBL7283113

SCHEMBL7283113

COC(=O)C=Cc1ccc(N2CCN(c3ccc(C#N)cc3)C2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 2/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
TYR P14679 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PTPN1 P18031 1/20 0.42
GPR183 P32249 1/20 0.41
P4HB P07237 1/20 0.41
TTR P02766 1/20 0.41
APP P05067 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PRMT1 Q99873 1/20 0.40
SNCA P37840 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283110 1.00 HDAC2 (0.48) HDAC2CA12CA1CA2TYR
SCHEMBL7102981 0.84 CA12 (0.64) HDAC2CA12CA1CA2TYR
SCHEMBL7102972 0.84 CA12 (0.64) HDAC2CA12CA1CA2TYR
SCHEMBL7272534 0.81 HDAC2 (0.49) HDAC2CA12CA1CA2TYR
SCHEMBL7272529 0.81 HDAC2 (0.49) HDAC2CA12CA1CA2TYR
Oxirane SCHEMBL28643072 0.80 CA12 (0.55) HDAC2CA12CA1CA2TYR
SCHEMBL13114501 0.80 HDAC2 (0.68) HDAC2CA12CA1CA2TYR
Hydrochloric Acid SCHEMBL7284305 0.79 F10 (0.48) CA12CA1CA2TYRCA7
Hydrochloric Acid SCHEMBL8911680 0.79 F10 (0.48) CA12CA1CA2TYRCA7
SCHEMBL7393580 0.77 CA12 (0.51) HDAC2CA12CA1CA2TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed