SCHEMBL7283243

SCHEMBL7283243

COC(=O)CCc1ccc(N2CCN(c3ccc(CCN)cc3)C2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.44
S1PR1 P21453 1/20 0.43
HDAC1 Q13547 3/20 0.41
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
EPHX2 P34913 1/20 0.39
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
MAPT P10636 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
TP53 P04637 1/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
IDO1 P14902 1/20 0.37
CTSG P08311 1/20 0.37
CMA1 P23946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281838 0.92 HRH3 (0.44) HRH3S1PR1HDAC1EPHX2ADRB2
Hydrochloric Acid SCHEMBL7282229 0.91 HRH3 (0.43) HRH3S1PR1HDAC1EPHX2ADRB2
Hydrochloric Acid SCHEMBL8910783 0.90 SIRT2 (0.40) HRH3S1PR1HDAC1ITGB3ITGA2B
SCHEMBL7282587 0.90 CYP4F2 (0.50) S1PR1HDAC1ITGB3ITGA2BMAPT
Propylamine SCHEMBL8911200 0.89 S1PR1 (0.44) HRH3S1PR1HDAC1MAPTCYP4F2
SCHEMBL27397736 0.88 MEN1 (0.51) HRH3S1PR1HDAC1TP53CTSG
Hydrochloric Acid SCHEMBL7272819 0.86 HRH3 (0.44) HRH3S1PR1HDAC1EPHX2ADRB2
SCHEMBL7280993 0.86 HDAC1 (0.46) HRH3S1PR1HDAC1MAPT
SCHEMBL7283131 0.86 HRH3 (0.43) HRH3S1PR1HDAC1EPHX2ADRB2
SCHEMBL7272906 0.86 F10 (0.42) HRH3S1PR1HDAC1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed