SCHEMBL7283891

SCHEMBL7283891

Cc1cc(C=O)c(OCC=CCOc2c(C=O)cc(C)cc2C=O)c(C=O)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.50
ERN1 O75460 2/20 0.47
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 10/20 0.34
LMNA P02545 3/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 2/20 0.32
TSHR P16473 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
MPI P34949 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.31
TUBB1 Q9H4B7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283882 1.00 SRC (0.50) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL7284734 0.82 SRC (0.52) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL7283876 0.80 SRC (0.50) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL6736649 0.78 SRC (0.49) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL7290764 0.77 SRC (0.47) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL28464657 0.77 ERN1 (0.44) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL6737227 0.74 ERN1 (0.57) SRCERN1NPSR1ALDH1A1LMNA
SCHEMBL4298275 0.74 KMT2A (0.40) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL4298273 0.74 KMT2A (0.40) ALDH1A1KDM4EMAPTL3MBTL1MEN1
SCHEMBL9146840 0.73 SRC (0.44) SRCERN1NPSR1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656362-B1 Macrocyclic compounds and their use as pharmaceuticals LILLY CO ELI (GB) 1999-09-01 EP disclosed
US-5580900-A TREATMENT OF DISEASES OF CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1996-12-03 US disclosed
US-5574158-A CRYPT COMPOUNDS, NERVOUS SYSTEM DISORDERS, CHELATE COMPOUNDS LILLY INDUSTRIES LIMITED (GB) 1996-11-12 US disclosed
EP-0656362-A1 Novel compounds LILLY INDUSTRIES LIMITED (GB) 1995-06-07 EP disclosed