SCHEMBL7286279

SCHEMBL7286279

CC(C)C(NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)c1ncco1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 3/20 0.51
ELANE P08246 13/20 0.51
CMA1 P23946 1/20 0.50
MALT1 Q9UDY8 1/20 0.48
CCR1 P32246 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13814740 0.84 ELANE (0.53) CAPN1ELANECMA1MALT1
SCHEMBL7278810 0.84 ELANE (0.52) CAPN1ELANECMA1MALT1CCR1
SCHEMBL10081595 0.82 ELANE (0.65) ELANECMA1
SCHEMBL10081596 0.81 ELANE (0.57) CAPN1ELANECMA1
SCHEMBL17425092 0.81 CMA1 (0.56) CAPN1ELANECMA1CCR1
SCHEMBL1506200 0.81 ALDH1A1 (0.62) CAPN1ELANECMA1CCR1
SCHEMBL22209363 0.81 ALDH1A1 (0.62) CAPN1ELANECMA1CCR1
SCHEMBL30051146 0.81 ALDH1A1 (0.62) CAPN1ELANECMA1CCR1
SCHEMBL1506251 0.81 ACE (0.61) CAPN1ELANECMA1CCR1
SCHEMBL10063674 0.81 ACE (0.61) CAPN1ELANECMA1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0291234-B1 Peptidic human leukocyte elastase (HLE) inhibitors ZENECA INC (US) 1994-03-23 EP disclosed
US-5164371-A HETEROCYCLIC KETONES ICI AMERICAS INC. (US) 1992-11-17 US disclosed
EP-0291234-A2 Peptidic human leukocyte elastase (HLE) inhibitors ZENECA INC. (US) 1988-11-17 EP disclosed