SCHEMBL7287145

SCHEMBL7287145

COc1cccc(CCCCc2c(CC#N)ccc(OC)c2OC)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.53
ABCB1 P08183 5/20 0.46
ABCG2 Q9UNQ0 1/20 0.44
ACHE P22303 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
BCHE P06276 3/20 0.43
TAAR1 Q96RJ0 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7295345 0.98 SLC2A1 (0.53) SLC2A1ABCB1ABCG2ACHECHRM2
SCHEMBL7283720 0.93 SLC2A1 (0.58) SLC2A1ABCB1ABCG2CHRM2CHRM1
SCHEMBL7293467 0.84 SLC2A1 (0.56) SLC2A1ABCB1ABCG2ACHECHRM2
SCHEMBL7286452 0.83 SLC2A1 (0.45) SLC2A1ABCB1ABCG2TAAR1
Hydrochloric Acid SCHEMBL7292452 0.82 SLC2A1 (0.60) SLC2A1ABCB1ABCG2ACHETAAR1
SCHEMBL7293616 0.82 SLC2A1 (0.56) SLC2A1ABCB1ABCG2ACHECHRM2
SCHEMBL7285836 0.82 KDM4E (0.48) SLC2A1ABCB1ABCG2
Hydrochloric Acid SCHEMBL7292865 0.80 SLC2A1 (0.60) SLC2A1ABCB1ABCG2CHRM2CHRM1
SCHEMBL7285255 0.80 SLC2A1 (0.47) SLC2A1ABCB1ACHETAAR1
SCHEMBL7279399 0.79 SLC2A1 (0.49) SLC2A1ABCB1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223598-B1 CATECHOLAMINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF FISONS plc (GB) 1991-06-12 EP disclosed
US-4939147-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC. (GB) 1990-07-03 US disclosed
US-4922022-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC (GB) 1990-05-01 US disclosed
US-4883804-A Aromatic compounds FISONS PLC (GB) 1989-11-28 US disclosed
EP-0223598-A2 Catecholamine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-05-27 EP disclosed