SCHEMBL7288263

SCHEMBL7288263

Cc1ccc(CC2(O)CCN(C(C)COc3ccc(O)cc3)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 8/20 0.65
GRIN2D O15399 5/20 0.65
GRIN3B O60391 5/20 0.65
GRIN1 Q05586 5/20 0.65
GRIN2A Q12879 5/20 0.65
GRIN2C Q14957 5/20 0.65
GRIN3A Q8TCU5 5/20 0.65
MAPT P10636 1/20 0.65
ADRA1A P35348 4/20 0.54
ADRA1D P25100 2/20 0.54
ADRA1B P35368 2/20 0.54
GAA P10253 1/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
OPRL1 P41146 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7295429 0.99 GRIN2B (0.64) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7290028 0.82 GRIN2B (0.73) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL7294297 0.81 GRIN2B (0.72) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7289795 0.81 GAA (0.68) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL499394 0.79 GRIN2D (1.00) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL1994218 0.78 GRIN2D (0.98) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9963240 0.77 GRIN2B (0.54) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8485641 0.72 GRIN2B (0.53) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL7287517 0.72 GRIN2B (0.51) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7294333 0.72 TSHR (0.62) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824098-B1 4-hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-10-31 EP claimed
EP-0824098-A1 4-hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-02-18 EP claimed
EP-0824098-B1 4-hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-10-31 EP disclosed
US-5889026-A 4-hydroxy-piperodine derivatives HOFFMANN-LA ROCHE INC. (US) 1999-03-30 US disclosed
EP-0824098-A1 4-hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-02-18 EP disclosed