SCHEMBL7288808

SCHEMBL7288808

COc1ccccc1OCC(O)CN1CCN(CC(=O)Nc2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.67
TSHR P16473 3/20 0.67
CYP2D6 P10635 2/20 0.67
NFKB1 P19838 1/20 0.67
ADRB2 P07550 1/20 0.67
ADRB1 P08588 1/20 0.67
ADRA2A P08913 1/20 0.67
ADRA2B P18089 1/20 0.67
ADRA2C P18825 1/20 0.67
ADRA1A P35348 1/20 0.67
DRD3 P35462 1/20 0.67
HTR2B P41595 1/20 0.67
KCNH2 Q12809 1/20 0.67
SCN5A Q14524 1/20 0.67
LMNA P02545 4/20 0.66
NPSR1 Q6W5P4 2/20 0.66
BLM P54132 1/20 0.66
PMP22 Q01453 1/20 0.66
ALDH1A1 P00352 6/20 0.58
KMT2A Q03164 4/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279229 0.90 TSHR (0.72) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7289216 0.89 TSHR (0.71) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7283156 0.89 TSHR (0.70) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7279519 0.87 CYP3A4 (0.76) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7291659 0.87 CYP2D6 (0.76) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7282209 0.86 CYP3A4 (0.72) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7288559 0.86 CYP3A4 (0.72) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7292174 0.86 TSHR (0.72) CYP3A4TSHRCYP2D6NFKB1ADRB2
SCHEMBL7288487 0.86 TSHR (0.72) CYP3A4TSHRCYP2D6NFKB1ADRB2
Hydrochloric Acid SCHEMBL7300686 0.86 LMNA (0.76) CYP3A4TSHRCYP2D6NFKB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed