SCHEMBL7290004

SCHEMBL7290004

COc1ccc2c(c1)C[C@H](C(=O)O)O2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.57
GABRA1 P14867 2/20 0.55
GABRB2 P47870 2/20 0.55
MTNR1A P48039 3/20 0.51
PPARD Q03181 1/20 0.51
HRH3 Q9Y5N1 2/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ABCB1 P08183 1/20 0.47
AR P10275 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
LMNA P02545 2/20 0.45
TP53 P04637 1/20 0.44
CYP19A1 P11511 1/20 0.44
MAOB P27338 1/20 0.44
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7289411 1.00 GLS (0.57) GLSGABRA1GABRB2MTNR1APPARD
SCHEMBL7289417 1.00 GLS (0.57) GLSGABRA1GABRB2MTNR1APPARD
SCHEMBL7286847 0.88 GLS (0.46) GLSGABRA1GABRB2MTNR1APPARD
SCHEMBL7286852 0.88 GLS (0.46) GLSGABRA1GABRB2MTNR1APPARD
SCHEMBL29443014 0.87 GLS (0.56) GLSGABRA1GABRB2MTNR1AHRH3
SCHEMBL4455342 0.87 GLS (0.56) GLSGABRA1GABRB2MTNR1AHRH3
SCHEMBL7296319 0.85 PPARG (0.51) GLSGABRA1GABRB2MTNR1AMEN1
SCHEMBL7296313 0.85 PPARG (0.51) GLSGABRA1GABRB2MTNR1AMEN1
SCHEMBL24193318 0.80 TDP1 (0.46) GLSKMT2APOLBCYP3A4CYP2C9
SCHEMBL14546592 0.79 KDM4E (0.48) GLSPPARDALDH1A1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6359138-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2002-03-19 US disclosed
EP-0846683-B1 4-Hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-09-19 EP disclosed
EP-0846683-A1 4-Hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-06-10 EP disclosed