SCHEMBL7291746

SCHEMBL7291746

CCOC(=O)c1c[nH]c2c(OC)ccc(-c3ccccc3)c2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLEC4M Q9H2X3 1/20 0.51
KDM4E B2RXH2 3/20 0.46
JAK2 O60674 3/20 0.46
JAK3 P52333 3/20 0.46
MAPT P10636 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
GABRA1 P14867 3/20 0.44
GABRB2 P47870 3/20 0.44
GABRB1 P18505 2/20 0.44
GABRA3 P34903 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
PPARG P37231 1/20 0.43
HTT P42858 1/20 0.41
CDC25B P30305 1/20 0.41
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829849 0.86 CLEC4M (0.56) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL7291947 0.83 CLEC4M (0.54) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL62162 0.81 CLEC4M (0.52) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL7291074 0.77 CLEC4M (0.50) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL397393 0.77 CLEC4M (0.52) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL774558 0.76 CLEC4M (0.76) CLEC4MKDM4EMAPTCYP1A2CYP3A4
SCHEMBL14845114 0.75 CLEC4M (0.63) CLEC4MKDM4EMAPTCYP1A2CYP3A4
SCHEMBL7290870 0.75 CLEC4M (0.63) CLEC4MKDM4EMAPTCYP1A2CYP3A4
SCHEMBL320357 0.74 TSHR (0.53) CLEC4MKDM4EJAK2JAK3MAPT
SCHEMBL396665 0.74 CLEC4M (0.57) CLEC4MKDM4EMAPTGABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0343574-B1 4(1H)-quinolone derivatives KIRIN BREWERY (JP) 1994-07-27 EP claimed
EP-0343574-B1 4(1H)-quinolone derivatives KIRIN BREWERY (JP) 1994-07-27 EP disclosed
US-5081121-A Cardiotonic agents KIRIN BEER KABUSHIKI KAISHA (JP) 1992-01-14 US disclosed
EP-0343574-A1 4(1H)-quinolone derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1989-11-29 EP disclosed