SCHEMBL7293124

SCHEMBL7293124

CS(=O)(=O)Nc1ccc2[nH]c(=O)n(CCCCN3CC=C(c4ccccc4)CC3)c(=O)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.50
KDM4E B2RXH2 3/20 0.49
TDP1 Q9NUW8 3/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HSD17B10 Q99714 3/20 0.49
TSHR P16473 2/20 0.49
ALOX15 P16050 2/20 0.49
USP2 O75604 1/20 0.49
HTT P42858 1/20 0.49
HTR1A P08908 2/20 0.43
NPC1 O15118 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7296451 0.99 PARP1 (0.49) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7299614 0.93 KDM4E (0.49) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7287843 0.92 PARP1 (0.49) PARP1KDM4ETDP1ALDH1A1MAPT
Sulfuric Acid SCHEMBL7329510 0.90 KDM4E (0.49) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7297124 0.88 PARP1 (0.53) PARP1KDM4ETDP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7301692 0.84 PARP1 (0.56) PARP1
SCHEMBL7292780 0.83 PARP1 (0.55) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7298716 0.83 PARP1 (0.58) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7297348 0.82 KDM4E (0.49) PARP1KDM4ETDP1ALDH1A1MAPT
SCHEMBL7300024 0.82 PARP1 (0.58) PARP1KDM4ETDP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436157-B1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-23 EP claimed
US-5296487-A Dopamine antagonist for nervous system disorders FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US claimed
US-5264438-A Dopamine receptor agonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-11-23 US claimed
EP-0436157-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-07-10 EP claimed
JP-5078349-A None JP disclosed
EP-0436157-B1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-23 EP disclosed
US-5296487-A Dopamine antagonist for nervous system disorders FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
US-5264438-A Dopamine receptor agonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-11-23 US disclosed
WO-1993018769-A2 A NEW USE OF QUINAZOLINE DERIVATIVE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-09-30 WO disclosed
JP-H0578349-A QUINAZOLINE DERIVATIVE AND ITS PRODUCTION FUJISAWA PHARMACEUT CO LTD 1993-03-30 JP disclosed
EP-0436157-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-07-10 EP disclosed