SCHEMBL7293158

SCHEMBL7293158

CCOC(=O)N(C(C)=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
HSD17B10 Q99714 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
HPGD P15428 1/20 0.49
CTDSP1 Q9GZU7 1/20 0.49
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
POLB P06746 2/20 0.46
LMNA P02545 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP3A4 P08684 1/20 0.46
TSHR P16473 2/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
GAA P10253 2/20 0.43
MDM2 Q00987 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5933087 0.87 ALDH1A1 (0.51) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL5933074 0.86 ALDH1A1 (0.49) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL3781111 0.86 ALDH1A1 (0.49) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL11688083 0.84 ALDH1A1 (0.48) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL5933048 0.84 ALDH1A1 (0.51) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL5933058 0.84 ALDH1A1 (0.48) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL10869589 0.84 ALDH1A1 (0.48) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL24340465 0.83 ALDH1A1 (0.58) ALDH1A1MAPTHPGDKMT2ALMNA
SCHEMBL27382574 0.83 ALDH1A1 (0.47) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9
SCHEMBL11211446 0.81 ALDH1A1 (0.46) ALDH1A1MAPTHSD17B10CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449346-B1 4-Piperidinyl-ergoline derivatives PHARMACIA SPA (IT) 1995-05-10 EP disclosed
EP-0449346-A2 4-Piperidinyl-ergoline derivatives PHARMACIA S.p.A. (IT) 1991-10-02 EP disclosed