SCHEMBL7293178

SCHEMBL7293178

CC(C)C(C(N)=O)N(Cc1ccncc1)C(=O)C(Cc1ccccc1)CC(O)C(Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.56
PSEN1 P49768 3/20 0.55
PSEN2 P49810 3/20 0.55
APH1B Q8WW43 3/20 0.55
NCSTN Q92542 3/20 0.55
APH1A Q96BI3 3/20 0.55
PSENEN Q9NZ42 3/20 0.55
APP P05067 1/20 0.55
KLK5 Q9Y337 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299783 0.95 PSEN1 (0.59) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7301635 0.90 PSEN1 (0.54) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7296543 0.89 PSEN1 (0.53) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7301983 0.87 PSEN1 (0.57) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7293457 0.85 PSEN1 (0.56) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7299761 0.85 PSEN1 (0.56) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7301536 0.83 PSEN1 (0.54) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7292722 0.82 PSEN1 (0.51) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7302349 0.82 PSEN1 (0.51) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL7302103 0.81 PSEN1 (0.54) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337714-A2 HIV protease inhibitors useful for the treatment of aids MERCK & CO. INC. (US) 1989-10-18 EP claimed