SCHEMBL7294375

SCHEMBL7294375

CN(C(=O)c1ccccc1)c1cccc(O[C]=O)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 9/20 0.56
HSD17B1 P14061 8/20 0.56
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HTT P42858 1/20 0.44
KDM1A O60341 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
PLAU P00749 1/20 0.44
TSHR P16473 1/20 0.43
ATM Q13315 1/20 0.43
NR1H3 Q13133 2/20 0.42
NR1H2 P55055 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001629 0.81 KMT2A (0.62) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL7294383 0.80 HSD17B2 (0.56) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL14878168 0.78 KMT2A (0.61) HSD17B2HSD17B1KMT2AKDM4ETSHR
SCHEMBL4181087 0.77 KMT2A (0.57) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL3185124 0.76 BCHE (0.46) HSD17B2HSD17B1TSHR
SCHEMBL493114 0.76 KMT2A (0.75) KMT2AKDM4EHTTKDM1AMAOA
SCHEMBL10212283 0.75 HSD17B2 (0.72) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL18780858 0.75 KMT2A (0.56) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL29940968 0.75 HSD17B2 (0.72) HSD17B2HSD17B1KMT2AKDM4EHTT
SCHEMBL12495904 0.75 HSD17B2 (0.90) HSD17B2HSD17B1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed
EP-0382185-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed