SCHEMBL7294657

SCHEMBL7294657

COc1cccc(CCNC(=O)CCCCC(=O)O)c1

nearest known ligand 0.79

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
MTNR1A P48039 1/20 0.63
MTNR1B P49286 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
EPHX2 P34913 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30639518 0.92 KMT2A (0.65) MTNR1AMTNR1BMEN1KMT2A
Hydrochloric Acid SCHEMBL30639528 0.91 KMT2A (0.64) MTNR1AMTNR1BMEN1KMT2A
SCHEMBL21449764 0.90 MEN1 (0.72) HDAC1HDAC6MTNR1AMTNR1BMEN1
SCHEMBL27419965 0.90 EPHX2 (0.75) MTNR1AMTNR1BEPHX2
SCHEMBL17283413 0.89 EPHX2 (0.77) HDAC1HDAC6MTNR1AMTNR1BEPHX2
SCHEMBL3199590 0.87 MTNR1A (0.62) HDAC1HDAC6MTNR1AMTNR1BSMN1; SMN2
SCHEMBL1665670 0.86 MTNR1A (0.61) MTNR1AMTNR1BMEN1KMT2A
SCHEMBL23026415 0.85 HDAC1 (0.61) HDAC1HDAC6MTNR1AMTNR1BEPHX2
SCHEMBL29722609 0.85 MTNR1A (0.67) MTNR1AMTNR1BEPHX2
SCHEMBL24528927 0.85 MTNR1A (0.67) MTNR1AMTNR1BEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223598-B1 CATECHOLAMINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF FISONS plc (GB) 1991-06-12 EP disclosed
US-4939147-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC. (GB) 1990-07-03 US disclosed
US-4922022-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC (GB) 1990-05-01 US disclosed
US-4883804-A Aromatic compounds FISONS PLC (GB) 1989-11-28 US disclosed
EP-0223598-A2 Catecholamine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-05-27 EP disclosed