SCHEMBL7295304

SCHEMBL7295304

O=C(OC1CC2CCC(C1)N2)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.63
HTR3E A5X5Y0 1/20 0.61
GMNN O75496 1/20 0.61
HTR3B O95264 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
ALOX15 P16050 1/20 0.61
TSHR P16473 1/20 0.61
MTOR P42345 1/20 0.61
HTR3A P46098 1/20 0.61
PMP22 Q01453 1/20 0.61
HTR3D Q70Z44 1/20 0.61
HTR3C Q8WXA8 1/20 0.61
HSD17B10 Q99714 1/20 0.61
GAA P10253 1/20 0.59
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
POLB P06746 1/20 0.50
SLC6A4 P31645 3/20 0.44
SLC6A2 P23975 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302350 0.81 CHRNA7 (0.63) CHRNA7HTR3EGMNNHTR3BCYP1A2
SCHEMBL1103724 0.78 CHRNA7 (1.00) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL221269 0.78 CHRNA7 (1.00) CHRNA7HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL195148 0.76 CYP2D6 (1.00) CHRNA7HTR3EGMNNHTR3BCYP1A2
Bemesetron SCHEMBL10765684 0.76 CYP2D6 (1.00) CHRNA7HTR3EGMNNHTR3BCYP1A2
Bemesetron SCHEMBL5790539 0.76 CYP2D6 (1.00) CHRNA7HTR3EGMNNHTR3BCYP1A2
Bemesetron SCHEMBL195147 0.76 CYP2D6 (1.00) CHRNA7HTR3EGMNNHTR3BCYP1A2
Bemesetron SCHEMBL29430183 0.76 CYP2D6 (1.00) CHRNA7HTR3EGMNNHTR3BCYP1A2
SCHEMBL31544490 0.73 KMT2A (0.81) CHRNA7CYP1A2CYP2D6TSHRMEN1
SCHEMBL31544489 0.73 KMT2A (0.81) CHRNA7CYP1A2CYP2D6TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090076019-A1 METHODS FOR TREATING NEUROLOGICAL DISORDERS OR DAMAGE MOUNT SINAI HOSPITAL (CA) 2009-03-19 US disclosed
US-5252570-A Amidino and guanidino derivatives B.I. ITALIA (IT) 1993-10-12 US disclosed
US-5047410-A Indolyl derivatives and their use as 5-HT3, receptor antagonists ISTITUTO DE ANGELI S.P.A. (IT) 1991-09-10 US disclosed
EP-0351385-A2 New amidino and guanidino derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-01-17 EP disclosed