SCHEMBL7302350

SCHEMBL7302350

Cc1cc(C)cc(C(=O)OC2CC3CCC(C2)N3)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.63
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2D6 P10635 2/20 0.62
HTR3E A5X5Y0 2/20 0.62
HTR3B O95264 2/20 0.62
HTR3A P46098 2/20 0.62
HTR3D Q70Z44 2/20 0.62
HTR3C Q8WXA8 2/20 0.62
CYP2C19 P33261 1/20 0.62
NR1I2 O75469 1/20 0.62
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
GMNN O75496 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
MTOR P42345 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7295304 0.81 CHRNA7 (0.63) CHRNA7MEN1KMT2ACYP1A2CYP2D6
SCHEMBL221269 0.78 CHRNA7 (1.00) CHRNA7MEN1KMT2AHTR3EHTR3B
SCHEMBL7301448 0.78 CYP2D6 (0.57) MEN1KMT2ACYP1A2CYP2D6HTR3E
SCHEMBL1103724 0.78 CHRNA7 (1.00) CHRNA7MEN1KMT2AHTR3EHTR3B
Tropanserin SCHEMBL467253 0.77 CYP2D6 (1.00) CHRNA7MEN1KMT2ACYP1A2CYP2D6
Tropanserin SCHEMBL29385911 0.77 CYP2D6 (1.00) CHRNA7MEN1KMT2ACYP1A2CYP2D6
SCHEMBL27815808 0.77 MEN1 (0.60) MEN1KMT2ACYP1A2CYP2D6HTR3E
Hydrochloric Acid SCHEMBL7301306 0.76 KMT2A (0.56) MEN1KMT2ACYP1A2CYP2D6HTR3E
Tropanserin SCHEMBL29400878 0.76 CYP2D6 (0.97) CHRNA7MEN1KMT2ACYP1A2CYP2D6
SCHEMBL31544490 0.76 KMT2A (0.81) CHRNA7MEN1KMT2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252570-A Amidino and guanidino derivatives B.I. ITALIA (IT) 1993-10-12 US disclosed
EP-0351385-A2 New amidino and guanidino derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-01-17 EP disclosed