SCHEMBL7295404

SCHEMBL7295404

COc1cc(NC(=O)c2ccc(C(C)(C)C)cc2)ccc1C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.67
SMN1; SMN2 Q16637 5/20 0.67
TP53 P04637 4/20 0.67
MAPT P10636 4/20 0.67
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
LMNA P02545 2/20 0.61
MAPK1 P28482 1/20 0.61
ATM Q13315 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
ALDH1A1 P00352 1/20 0.58
PPARG P37231 1/20 0.57
PPARA Q07869 1/20 0.57
HDAC3 O15379 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
KCNK9 Q9NPC2 1/20 0.56
THRB P10828 1/20 0.55
GRM4 Q14833 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9696412 0.89 NR1H4 (0.77) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL95373 0.84 NPC1 (0.59) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL14347581 0.84 KMT2A (0.74) SMN1; SMN2TP53MAPTNPC1RAB9A
SCHEMBL7301385 0.84 NPC1 (0.69) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL7301440 0.82 SMN1; SMN2 (0.78) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL7295519 0.80 NPC1 (0.66) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL21588673 0.80 HDAC6 (0.67) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL25721410 0.80 HDAC6 (0.67) NR1H4SMN1; SMN2TP53MAPTNPC1
SCHEMBL7303163 0.78 HDAC3 (0.86) NR1H4SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL9447193 0.78 CYP1A2 (0.56) MAPTLMNAALDH1A1GRM4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358118-B1 Phenylamides - process for their preparation as well as a drug containing those compounds BOEHRINGER MANNHEIM GMBH (DE) 1994-03-16 EP disclosed
US-5135949-A Anticoagulants BOEHRINGER MANNHEIM GMBH (DE) 1992-08-04 US disclosed
EP-0358118-A1 Phenylamides - process for their preparation as well as a drug containing those compounds Roche Diagnostics GmbH (DE) 1990-03-14 EP disclosed