SCHEMBL7298577

SCHEMBL7298577

[O]c1cc(Cl)cc2cccc(Cl)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
ALDH1A1 P00352 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP2A6 P11509 3/20 0.37
CYP1A2 P05177 2/20 0.37
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
AHR P35869 2/20 0.34
DAO P14920 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
DOT1L Q8TEK3 1/20 0.33
PARP1 P09874 1/20 0.33
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14375274 0.82 AHR (0.42) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL18242843 0.78 MEN1 (0.46) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL8723829 0.75 CYP2A6 (0.37) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL5255668 0.75 AHR (0.37) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL5255665 0.75 CYP2A6 (0.37) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL8723827 0.75 CYP2A6 (0.37) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL29344202 0.75 CYP2A6 (0.37) MEN1KMT2AALDH1A1RXFP1KDM4E
SCHEMBL2362910 0.72 ALDH1A1 (0.61) MEN1KMT2AALDH1A1KDM4ETSHR
SCHEMBL15351928 0.70 CYP2A6 (0.44) MEN1KMT2AALDH1A1KDM4ETSHR
SCHEMBL29620230 0.69 TSHR (0.53) MEN1KMT2AALDH1A1RXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed