SCHEMBL7298902

SCHEMBL7298902

FC(F)(F)C1=NCCc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.53
NOS2 P35228 1/20 0.53
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAOA P21397 2/20 0.40
CES1 P23141 1/20 0.38
CYP19A1 P11511 4/20 0.35
CYP11B2 P19099 3/20 0.35
CYP11B1 P15538 2/20 0.35
CYP2A6 P11509 1/20 0.34
MAOB P27338 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
TSHR P16473 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29964099 1.00 NOS3 (0.53) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL11778063 0.85 NOS3 (0.50) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL11779898 0.82 NOS3 (0.47) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL14001394 0.81 NOS3 (0.53) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL19794689 0.75 CYP19A1 (0.41) CYP19A1CYP11B2CYP11B1ADRA2A
SCHEMBL15399817 0.75 TDP1 (0.39) NOS3NOS2CYP19A1CYP11B2CYP11B1
SCHEMBL2796047 0.75 NOS3 (0.47) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL3056563 0.73 NOS3 (0.45) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL29361631 0.71 KDM4E (0.60) NOS3NOS2KDM4EALDH1A1MAOA
SCHEMBL7509399 0.71 KDM4E (0.60) NOS3NOS2KDM4EALDH1A1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11161102-B2 Iminium salt organocatalysts, method of making, and methods of using UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2021-11-02 US disclosed
US-11161102-B2 Iminium salt organocatalysts, method of making, and methods of using UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2021-11-02 US disclosed
US-20190344253-A1 IMINIUM SALT ORGANOCATALYSTS, METHOD OF MAKING, AND METHODS OF USING UNIV VIRGINIA PATENT FOUNDATION (US) 2019-11-14 US disclosed
US-20190344253-A1 IMINIUM SALT ORGANOCATALYSTS, METHOD OF MAKING, AND METHODS OF USING UNIV VIRGINIA PATENT FOUNDATION (US) 2019-11-14 US disclosed
WO-2017223287-A1 IMINIUM SALT ORGANOCATALYSTS, METHODS OF MAKING, AND METHODS OF USING UNIVERSITY OF VIRGINIA (US) 2017-12-28 WO disclosed
US-5605926-A PROPHYLAXIS BAYER AKTIENGESELLSCHAFT (DE) 1997-02-25 US disclosed
US-5430151-A Treatment of aids, pneumonia, caprine arthritis encephalitis, leukemia and immmunodeficiency BAYER AKTIENGESELLSCHAFT (DE) 1995-07-04 US disclosed
US-5204471-A α-trifluoromethyl-substituted, saturated bicyclic amines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed
EP-0527385-A1 Alpha-trifluoromethyl substituted, saturated bicyclic amines and process for their preparation BAYER AG (DE) 1993-02-17 EP disclosed