SCHEMBL7299441

SCHEMBL7299441

CC[C@H](NC(=O)N(C)Cc1ccccn1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.54
POLB P06746 2/20 0.44
MME P08473 1/20 0.44
PTPRA P18433 1/20 0.43
KCNK3 O14649 1/20 0.42
KCNA5 P22460 1/20 0.40
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LPAR1 Q92633 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27373122 1.00 CA2 (0.54) CA2POLBMMEPTPRAKCNK3
SCHEMBL27395775 0.84 CA2 (0.60) CA2POLBPTPRAKCNK3SMN1; SMN2
SCHEMBL7393135 0.84 CA2 (0.60) CA2POLBPTPRAKCNK3SMN1; SMN2
SCHEMBL7302427 0.84 CA2 (0.60) CA2POLBPTPRAKCNK3SMN1; SMN2
SCHEMBL4683895 0.83 CA2 (0.67) CA2POLBMMEPTPRASMN1; SMN2
SCHEMBL4683897 0.83 CA2 (0.67) CA2POLBMMEPTPRASMN1; SMN2
SCHEMBL7308111 0.79 CA2 (0.55) CA2KCNK3SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL27375082 0.79 HDAC1 (0.46) POLBMMEKDM4ELPAR1ALDH1A1
SCHEMBL7300357 0.79 HDAC1 (0.46) POLBMMEKDM4ELPAR1ALDH1A1
SCHEMBL2760067 0.78 CA2 (0.64) CA2POLBKCNK3SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0575097-B1 2,3-Bis-carboxamidomethyl substituted oxiranes as inhibitors of HIV protease and their use for the treatment of AIDS LILLY CO ELI (US) 2000-11-02 EP disclosed
US-5578608-A HIV PROTEASE INHIBITOR ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
EP-0575097-A1 2,3-Bis-carboxamidomethyl substituted oxiranes as inhibitors of HIV protease and their use for the treatment of AIDS ELI LILLY AND COMPANY (US) 1993-12-22 EP disclosed