SCHEMBL7299885

SCHEMBL7299885

CCOc1nc2cccc(OC(=O)OC(C)OC(=O)OC3CCCCC3)c2n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAE1 Q13564 4/20 0.69
AGTR2 P50052 3/20 0.69
PPARG P37231 3/20 0.69
CYP3A4 P08684 2/20 0.69
ADORA3 P0DMS8 2/20 0.69
ADRA2B P18089 2/20 0.69
SLC6A2 P23975 2/20 0.69
AGTR1 P30556 2/20 0.69
HTR2B P41595 2/20 0.69
PDE3A Q14432 2/20 0.69
KDM4E B2RXH2 1/20 0.69
MEN1 O00255 1/20 0.69
MLNR O43193 1/20 0.69
NR1I2 O75469 1/20 0.69
USP2 O75604 1/20 0.69
ESR1 P03372 1/20 0.69
NR3C1 P04150 1/20 0.69
TP53 P04637 1/20 0.69
PGR P06401 1/20 0.69
ADRB2 P07550 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Candesartan Cilexetil SCHEMBL1021483 0.92 NAE1 (0.79) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL16949997 0.92 NAE1 (0.79) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL40831 0.92 NAE1 (0.79) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL3968703 0.92 NAE1 (0.79) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL6515280 0.92 NAE1 (0.78) NAE1AGTR2PPARGCYP3A4ADORA3
SCHEMBL22198388 0.90 PPARG (0.63) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL474557 0.90 AGTR2 (0.76) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL1775074 0.89 NAE1 (0.75) NAE1AGTR2PPARGCYP3A4ADORA3
SCHEMBL14192229 0.89 PPARG (0.62) NAE1AGTR2PPARGCYP3A4ADORA3
Candesartan Cilexetil SCHEMBL1463446 0.89 AGTR2 (0.70) NAE1AGTR2PPARGCYP3A4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459136-B1 Benzimidazole derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-12-27 EP claimed