SCHEMBL7300067

SCHEMBL7300067

CCC(=O)c1cc([O])cc(C(=O)CC)c1C(=O)CC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.48
PTGS1 P23219 1/20 0.48
DRD3 P35462 1/20 0.48
HSP90AB1 P08238 1/20 0.44
HMGCR P04035 1/20 0.41
POLB P06746 1/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 3/20 0.34
CA9 Q16790 2/20 0.34
HSD17B10 Q99714 3/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.33
UBE2N P61088 1/20 0.33
TSHR P16473 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300081 0.82 MEN1 (0.65) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL8580424 0.80 MEN1 (0.47) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL7304067 0.73 KMT2A (0.43) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL18632252 0.71 MAPT (0.43) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL7308284 0.71 HSP90AB1 (0.47) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL7295691 0.70 HSP90AB1 (0.46) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL7193425 0.68 CYP3A4 (0.44) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL7308298 0.68 HSP90AB1 (0.37) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL13456583 0.67 HSP90AB1 (0.47) KMT2AMEN1CYP3A4PTGS1DRD3
SCHEMBL30918369 0.67 HSP90AB1 (0.47) KMT2AMEN1CYP3A4PTGS1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed