SCHEMBL7300176

SCHEMBL7300176

CC1(C)C=C(n2c(Cl)cccc2=O)c2ncccc2O1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
S100A4 P26447 1/20 0.30
CDC25B P30305 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7291851 0.81 MAPK14 (0.31) S100A4CDC25B
SCHEMBL7300272 0.78 NPC1 (0.33) NPC1
SCHEMBL7298971 0.77 CCNC (0.33) CDC25B
SCHEMBL7375797 0.77 NPC1 (0.32) NPC1
SCHEMBL7290451 0.77 CCNC (0.38)
SCHEMBL7368755 0.77 NPC1 (0.33) NPC1
SCHEMBL7370936 0.76 NPC1 (0.34) NPC1
SCHEMBL7313380 0.75 NPC1 (0.32) NPC1
SCHEMBL7369558 0.73 NPC1 (0.34) NPC1
SCHEMBL7294267 0.73 NPC1 (0.32) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308792-B1 AZACHROMANE DERIVATIVES MERCK PATENT GmbH (DE) 1993-07-28 EP disclosed
US-4931454-A Azachroman derivatives with effects on the cardiovascular system MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-06-05 US disclosed
EP-0308792-A2 Azachromane derivatives MERCK PATENT GmbH (DE) 1989-03-29 EP disclosed