SCHEMBL7300514

SCHEMBL7300514

c1ccc2c(c1)cc1n2CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.60
HTR2C P28335 5/20 0.60
SIGMAR1 Q99720 11/20 0.49
NOTUM Q6P988 1/20 0.43
HTR1A P08908 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18911620 1.00 HTR2A (0.60) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL29548539 0.98 HTR2A (0.62) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL669577 0.98 HTR2A (0.62) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL30703022 0.92 HTR2A (0.64) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL761931 0.92 HTR2A (0.64) HTR2AHTR2CSIGMAR1NOTUMHTR1A
Acetic Acid SCHEMBL13279290 0.87 HTR2A (0.55) HTR2AHTR2CSIGMAR1
SCHEMBL18911621 0.84 HTR2A (0.73) HTR2AHTR2CSIGMAR1NOTUMHTR1A
SCHEMBL7512405 0.76 KMT2A (0.54) NOTUMPOLB
SCHEMBL24916793 0.75 SIGMAR1 (0.50) HTR2AHTR2CSIGMAR1
SCHEMBL6711152 0.75 HTR2A (1.00) HTR2AHTR2CSIGMAR1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017088746-A1 NEW EPIDERMAL GROWTH FACTOR RECEPTOR INHIBITOR AND APPLICATION THEREOF 南京圣和药业股份有限公司 2017-06-01 WO disclosed
US-5721245-A ANTIINFLAMMATORY AGENTS, RESPIRATORY SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0384349-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1994-04-27 EP disclosed
US-5026696-A Psychotic disorders, anziety, nausea and vomiting GLAXO GROUP LIMITED (GB) 1991-06-25 US disclosed
US-4963546-A Ketone derivatives which are antagonists of 5-HT at 5-HT3 receptors, compositions containing them, and method of use GLAXO GROUP LIMITED (GB) 1990-10-16 US disclosed
EP-0384349-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1990-08-29 EP disclosed
EP-0327307-A2 Tricyclic ketone derivatives having a 5-HT3 antagonist activity GLAXO GROUP LIMITED (GB) 1989-08-09 EP disclosed