SCHEMBL7301124

SCHEMBL7301124

CC(C)(C)CC(=O)N[C@@H](Cc1ccccc1)C[C@H](O)[C@H](Cc1ccccc1)NC(=O)CC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.52
MME P08473 2/20 0.49
MMEL1 Q495T6 1/20 0.49
BCHE P06276 2/20 0.47
REN P00797 1/20 0.46
CA2 P00918 1/20 0.45
SLC6A11 P48066 1/20 0.44
CYP3A4 P08684 1/20 0.44
KLK5 Q9Y337 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309203 0.83 BACE1 (0.56) BACE1BCHERENSLC6A11
SCHEMBL7306950 0.81 BACE1 (0.63) BACE1BCHESLC6A11
SCHEMBL12294114 0.81 HPGD (0.59) MMEMMEL1
SCHEMBL8755186 0.81 HPGD (0.59) MMEMMEL1
SCHEMBL7305946 0.79 ATM (0.62) BACE1RENKLK5
SCHEMBL7270247 0.79 ATM (0.62) BACE1RENKLK5
SCHEMBL7299571 0.79 ATM (0.62) BACE1RENKLK5
SCHEMBL7301095 0.79 ATM (0.62) BACE1RENKLK5
SCHEMBL4957679 0.78 CA2 (0.43) BACE1MMEMMEL1BCHECA2
SCHEMBL4957683 0.78 CA2 (0.43) BACE1MMEMMEL1BCHECA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed