Acepromazine

Acepromazine

SCHEMBL73018

CC(=O)c1ccc2c(c1)N(CCCN(C)C)c1ccccc1S2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 11/20 1.00
CYP1A2 P05177 10/20 1.00
HTR1A P08908 7/20 1.00
DRD2 P14416 6/20 1.00
SLC6A2 P23975 6/20 1.00
SLC6A4 P31645 6/20 1.00
ADRA1A P35348 6/20 1.00
DRD3 P35462 6/20 1.00
KCNH2 Q12809 6/20 1.00
LMNA P02545 6/20 1.00
ADRA2A P08913 5/20 1.00
DRD1 P21728 5/20 1.00
CHRM2 P08172 5/20 1.00
CHRM1 P11229 5/20 1.00
SLC6A3 Q01959 5/20 1.00
TSHR P16473 4/20 1.00
OPRM1 P35372 4/20 1.00
PRNP P04156 3/20 1.00
TBXA2R P21731 2/20 1.00
TP53 P04637 5/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acepromazine SCHEMBL28142113 1.00 CYP2D6 (1.00) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL29582179 1.00 CYP2D6 (1.00) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL29441481 1.00 CYP2D6 (1.00) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL30620438 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL21803694 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL29876174 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL30616039 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL204733 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL7253707 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2
Acepromazine SCHEMBL204734 0.94 CYP2D6 (0.88) CYP2D6CYP1A2HTR1ADRD2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9976 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000641-A1 ISOTOPICALLY ENRICHED ANALOGS OF 5,6-METHYLENEDIOXY-2-AMINOINDANE (IMDAI) TERRAN BIOSCIENCES INC (US) 2026-01-01 US claimed
EP-4654963-A1 TREATMENT OF MENTAL ILLNESS VIA ADMINISTRATION OF BUNTANETAP AND ANALOGUES THEREOF Annovis Bio, Inc. (US) 2025-12-03 EP claimed
US-20250312353-A1 DRUG REPURPOSING FOR TREATMENT OF CONGENITAL VASCULAR MALFORMATIONS UNIVERSITY OF SOUTH CAROLINA (US) 2025-10-09 US claimed
US-12427140-B2 4-[5-[(rac)-1-[5-(3-chlorophenyl)-3-isoxazolyl]ethoxy]-4-methyl-4H-1,2,4-triazol-3-yl]pyridine for use in prevention and/or treatment of pain in an animal THULIN CLAES (SE) 2025-09-30 US claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250213647-A1 CHEMOKINE RECEPTORS AND ALPHA1 ADRENERGIC RECEPTORS/VASOPRESSIN RECEPTORS 1A HETEROMERS AS DRUG TARGETS FOR DISEASE UNIVERSITY OF SOUTH FLORIDA 2025-07-03 US claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
WO-2025101418-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. (US) 2025-05-15 WO claimed
US-20250144092-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. 2025-05-08 US claimed
EP-4547250-A1 METHODS AND COMPOSITIONS RELATING TO CONTROLLING PSYCHEDELIC EFFECTS WITH SEROTONIN RECEPTOR MODULATORS Terran Biosciences Inc. (US) 2025-05-07 EP claimed
WO-1993008801-A1 PREVENTION OF DRUG-INDUCED AGRANULOCYTOSIS WITH FREE RADICAL SCAVENGERS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-05-13 WO claimed
WO-1992021347-A1 IMPROVED EUTHANASIA COMPOSITIONS MICHIGAN STATE UNIVERSITY (US) 1992-12-10 WO claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
EP-0174342-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES. UNIV FLORIDA (US) 1986-03-19 EP claimed
WO-1985003937-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1985-09-12 WO claimed
US-4508715-A DOPAMINE ANTAGONISTS;OVERDOSE TREATMENT UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1985-04-02 US claimed
EP-0105361-A1 ANTAGONISM OF CENTRAL NERVOUS SYSTEM DRUGS BY THE ADMINISTRATION OF 4-AMINOPYRIDINE ALONE OR IN COMBINATION WITH OTHER DRUGS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1984-04-18 EP claimed
WO-1983003541-A1 ANTAGONISM OF CENTRAL NERVOUS SYSTEM DRUGS BY THE ADMINISTRATION OF 4-AMINOPYRIDINE ALONE OR IN COMBINATION WITH OTHER DRUGS UNIV GEORGIA RES FOUND (US) 1983-10-27 WO claimed
US-4249003-A Process for polycyclic amines AKTIEBOLAGET LEO (SE) 1981-02-03 US claimed
US-4213981-A ACEPROMAZINE AND MIDFLUR AMERICAN HOME PRODUCTS CORPORATION (US) 1980-07-22 US claimed